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Bis-alkylamine Indolo[3,2-b]quinolines as hemozoin ligands: implications for antimalarial cytostatic and cytocidal activities.
Structural optimization of quinolon-4(1H)-imines as dual-stage antimalarials: toward increased potency and metabolic stability.
Quinolin-4(1H)-imines are potent antiplasmodial drugs targeting the liver stage of malaria.
N-cinnamoylated chloroquine analogues as dual-stage antimalarial leads.
Enone- and chalcone-chloroquinoline hybrid analogues: in silico guided design, synthesis, antiplasmodial activity, in vitro metabolism, and mechanistic studies.
Incorporation of basic side chains into cryptolepine scaffold: structure-antimalarial activity relationships and mechanistic studies.
Design, synthesis, and development of novel guaianolide-endoperoxides as potential antimalarial agents.
Endoperoxide carbonyl falcipain 2/3 inhibitor hybrids: toward combination chemotherapy of malaria through a single chemical entity.
Falcipain inhibitors: optimization studies of the 2-pyrimidinecarbonitrile lead series.
Michael acceptor based antiplasmodial and antitrypanosomal cysteine protease inhibitors with unusual amino acids.