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Characterization of β-Carboline Derivatives Reveals a High Barrier to Resistance and Potent Activity against Ring-Stage and DHA-Induced Dormant Plasmodium falciparum.
Tambjamines as Fast-Acting Multistage Antimalarials.
Resistance to Some But Not Other Dimeric Lindenane Sesquiterpenoid Esters Is Mediated by Mutations in a Plasmodium falciparum Esterase.
Antimalarial Trioxolanes with Superior Drug-Like Properties and In Vivo Efficacy.